Raloxifene

Raloxifene is a selective estrogen receptor modulator (SERM) that works by binding to the estrogen receptors in the breast tissue, thereby preventing estrogen from binding to these receptors. This reduces the risk of gynecomastia and can even help reduce existing breast tissue.

Compared to Tamoxifen, Raloxifene has been shown to be more effective in reducing breast tissue in men with gynecomastia. Raloxifene is also less likely to cause side effects such as hot flashes and mood changes, making it a more tolerable option for bodybuilders.

When it comes to dosage, the optimal daily dose of Raloxifene for bodybuilders is typically 60-120mg per day. However, it is important to note that Raloxifene can have side effects, such as increased risk of blood clots and hot flashes, so it is important to speak with a healthcare provider before starting this medication.

In addition to its benefits for managing gynecomastia, Raloxifene has also been shown to have other benefits for bodybuilders. It can improve bone density, reduce the risk of cardiovascular disease, and even improve lipid profiles.